ACRALL

Nicotinic AcetylCholine Receptor Ligand Library

4,691 items of 157 Next page Last page

Name In Vivo Tested Phase Alpha4beta2 Alpha7 Muscletype PubChemCIDStructureMOL2File
TROPISETRON yes4antagonistpartial agonistUnknown activity
JNJ-39393406 yes4inactivePAM type Iinactive
Amantadine yes4N.A.NAMN.A.
NALTREXONE yes4antagonistNAMN.A.
buproprion yes4NAMNAMNAM
MECAMYLAMINE yes4NAMNAMNAM
ETOMIDATE yes4N.A.N.A.Unknown activity
1,10-Bis(trimethyl ammonium)decane dibromide yes4partial agonistN.A.N.A.
DECAMETHONIUM BROMIDE yes4partial agonistN.A.N.A.
succinylcholine yes4inactiveN.A.agonist
Galantamine yes4PAMinactiveinactive
Granisetron yes4inactiveinactiveN.A.
TUBOCURARINE CHLORIDE yes4antagonistantagonistN.A.
Tacrine yes4antagonistantagonistantagonist
Ondasetron yes4antagonistantagonistN.A.
CHOLINE yes4Unknown activityagonistUnknown activity
VARENICLINE yes4partial agonistagonistN.A.
ACETYLCHOLINE yes4agonistagonistagonist
Carbachol yes4agonistagonistN.A.
Carbamylcholine yes4agonistagonistagonist
NICOTINE yes4agonistagonistagonist
Encenicline yes3inactivepartial agonistinactive
Ivermectin yes3Unknown activityPAM type IN.A.
DEXMECAMYLAMINE yes3NAMNAMNAM
3,4-Methylenedioxymethamphetamine | MDMA yes3antagonistN.A.N.A.
DIANICLINE yes3partial agonistN.A.N.A.
CYTISINE yes3partial agonistagonistagonist
(-)-lobeline yes2Unknown activityUnknown activityUnknown activity
GTS-21 yes2inactivepartial agonistinactive
azd0328 yes2inactivepartial agonistinactive
Name In Vivo Tested Phase Alpha4beta2 Alpha7 Muscletype PubChemCIDStructureMOL2File
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